SB 706375
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0369
CAS Number: 733734-61-7
Purity: ≥98% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- Urotensin-ⅡReceptor
- CAS Number:
- 733734-61-7
- Chemical Name:
- 2-Bromo-4,5-dimethoxy-N-[3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]-4-(trifluoromethyl)phenyl]benzenesulfonamide
- Storage:
- Store at RT
- Molecular Formula:
- C20H22BrF3N2O5S
- Molecular Weight (kDa):
- 539.36
- Soluble:
- DMSO
Description
- Description:
- High affinity urotensin-Ⅱ receptor antagonist
Biological Activity
- Biological Activity:
- SB 706375 is a high affinity urotensin-Ⅱ receptor antagonist. It is non-peptide and can inhibit the binding of radiolabeled urotensin to endogenous human urotensin (UT) receptors.