SB 706375

SB 706375

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0369

CAS Number: 733734-61-7

Purity: ≥98% (HPLC)

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • Urotensin-ⅡReceptor
  • CAS Number:
  • 733734-61-7
  • Chemical Name:
  • 2-Bromo-4,5-dimethoxy-N-[3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]-4-(trifluoromethyl)phenyl]benzenesulfonamide
  • Storage:
  • Store at RT
  • Molecular Formula:
  • C20H22BrF3N2O5S
  • Molecular Weight (kDa):
  • 539.36
  • Soluble:
  • DMSO

Description

  • Description:
  • High affinity urotensin-Ⅱ receptor antagonist

Biological Activity

  • Biological Activity:
  • SB 706375 is a high affinity urotensin-Ⅱ receptor antagonist. It is non-peptide and can inhibit the binding of radiolabeled urotensin to endogenous human urotensin (UT) receptors.