Properties

• Target:
• CB1 Receptor

• CAS Number:
• 1998197-39-9

• Chemical Name:
• 6-methyl-3-(2-nitro-1-(thiophen-2-yl)ethyl)-2-phenyl-1H-indole

• Storage:
• Store at -20°C

• Molecular Formula:
• C21H18N2O2S

• Molecular Weight:
• 362.44

• Soluble:
• DMSO

Description

• Description:
• Positive allosteric modulator (PAM) of CB1 receptors

Biological Activity

• Biological Activity:
• ZCZ 011 is a brain penetrant positive allosteric modulator (PAM) of cannabinoid CB1 receptors. It can augment the pharmacological actions of the CB1 orthosteric agonists both _{in vitro} and _{in vivo}.