Properties

• Target:
• mGlu5 Receptor

• CAS Number:
• 871362-31-1

• Chemical Name:
• 2-chloro-4-((2,5-dimethyl-1-(4-(trifluoromethoxy)phenyl)-1H-imidazol-4-yl)ethynyl)pyridine

• Storage:
• Store at +4°C

• Molecular Formula:
• C19H13ClF3N3O

• Molecular Weight:
• 391.77

• Soluble:
• DMSO

Description

• Description:
• Potent and selective negative allosteric modulator (NAM) of mGlu5 receptors

Biological Activity

• Biological Activity:
• CTEP is a potent and selective negative allosteric modulator (NAM) of metabotropic glutamate receptor subtype 5 (mGluR5). It is orally bioavailable and long lasting.