Properties

• Target:
• TGR5

• CAS Number:
• 877052-79-4

• Chemical Name:
• 4-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-6-(2-fluorophenyl)-4,5-dihydro-pyrido[3,2-f]-1,4-oxazepin-3(2H)-one

• Storage:
• Store at -20°C

• Molecular Formula:
• C23H15F7N2O2

• Molecular Weight (kDa):
• 484.37

• Soluble:
• DMSO and Ethanol

Description

• Description:
• GPBA receptor (TGR5) agonist

Biological Activity

• Biological Activity:
• GPBAR-A is a GPBA receptor agonist. It can upregulate GLP-1 secretion from intestinal cultures.