Properties

• Target:
• GPER

• CAS Number:
• 881639-98-1

• Chemical Name:
• (±)-1-[(3aR*,4S*,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]- ethanone

• Storage:
• Store at -20°C

• Molecular Formula:
• C21H18BrNO3

• Molecular Weight (kDa):
• 412.28

• Soluble:
• DMSO

Description

• Description:
• Potent and selective GPER agonist

Biological Activity

• Biological Activity:
• G-1 is a potent and selective G-protein coupled estrogen receptor (GPER) agonist. It displays therapeutic effects in the mouse EAE model of multiple sclerosis.