GRI 977143

GRI 977143

For Research Use Only. Not For Clinical Use.

Catalog Number: AGO0222

CAS Number: 325850-81-5

Purity: ≥98% (HPLC)

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • LPA2 Receptor
  • CAS Number:
  • 325850-81-5
  • Chemical Name:
  • 2-[[3-(1,3-dioxo-1H-benz[de]isoquinolin-2(3H)-yl)propyl]thio]benzoic acid
  • Storage:
  • Store at +4°C
  • Molecular Formula:
  • C22H17NO4S
  • Molecular Weight (kDa):
  • 391.44
  • Soluble:
  • DMSO

Description

  • Description:
  • Selective LPA2 receptor non-lipid agonist

Biological Activity

  • Biological Activity:
  • GRI 977143 is a selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist. It can activate ERK1/2 survival pathway.