Properties

• Target:
• GPR39

• CAS Number:
• 1621175-65-2

• Chemical Name:
• N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide

• Storage:
• Store at +4°C

• Molecular Formula:
• C18H19ClN6O2S

• Molecular Weight (kDa):
• 418.9

• Soluble:
• DMSO

Description

• Description:
• Potent and selective GPR39 agonist

Biological Activity

• Biological Activity:
• TC-G 1008 is a potent and selective GPR39 agonist with oral bioavailability. It can increase GLP-1 levels in vitro and in vivo.