L-803,087 trifluoroacetate
For Research Use Only. Not For Clinical Use.
Catalog Number: AGO0336
CAS Number: 1786412-46-1
Purity: ≥97% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
Properties
- Target:
- SST4 Receptor
- CAS Number:
- 1786412-46-1
- Chemical Name:
- N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester trifluoroacetate
- Storage:
- Store at -20°C
- Molecular Formula:
- C25H29F2N5O3.CF3CO2H
- Molecular Weight (kDa):
- 599.56
- Soluble:
- DMSO and Ethanol
Description
- Description:
- Potent and selective SST4 receptor agonist
Biological Activity
- Biological Activity:
- L-803,087 trifluoroacetate is a potent and selective somatostatin SST4 receptor agonist. It can facilitate the hippocampal synaptic responses mediated by AMPA in vitro.