TBPB
For Research Use Only. Not For Clinical Use.
Catalog Number: ACT0004
CAS Number: 634616-95-8
Purity: 100%
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |

Properties
- Target:
- M1 Muscarinic Receptor
- CAS Number:
- 634616-95-8
- Chemical Name:
- 1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
- Storage:
- Store at +4°C
- Molecular Formula:
- C25H32N4O
- Molecular Weight (kDa):
- 404.55
- Soluble:
- DMSO
Description
- Description:
- Selective allosteric activator of the M1 muscarinic receptor
Biological Activity
- Biological Activity:
- TBPB is a selective allosteric activator of the M1 muscarinic receptor. In rodent models with antipsychotic-like activity, TBPB can increase the processing of non-amyloidogenic APP.