TBPB

TBPB

For Research Use Only. Not For Clinical Use.

Catalog Number: ACT0004

CAS Number: 634616-95-8

Purity: 100%

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • M1 Muscarinic Receptor
  • CAS Number:
  • 634616-95-8
  • Chemical Name:
  • 1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
  • Storage:
  • Store at +4°C
  • Molecular Formula:
  • C25H32N4O
  • Molecular Weight (kDa):
  • 404.55
  • Soluble:
  • DMSO

Description

  • Description:
  • Selective allosteric activator of the M1 muscarinic receptor

Biological Activity

  • Biological Activity:
  • TBPB is a selective allosteric activator of the M1 muscarinic receptor. In rodent models with antipsychotic-like activity, TBPB can increase the processing of non-amyloidogenic APP.