AM 281
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0108
CAS Number: 202463-68-1
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- CB1 Receptor
- CAS Number:
- 202463-68-1
- Chemical Name:
- 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide
- Storage:
- Desiccate at +4°C
- Molecular Formula:
- C21H19Cl2IN4O2
- Molecular Weight (kDa):
- 557.22
- Soluble:
- DMSO
Description
- Description:
- Potent and selective CB1 receptor antagonist
Biological Activity
- Biological Activity:
- AM 281 is a potent and selective CB1 receptor antagonist.Following systemic administration in vivo, it can increase locomotor activity.