CI 988
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0153
CAS Number: 130332-27-3
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- CCK2 Receptor
- CAS Number:
- 130332-27-3
- Chemical Name:
- 4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid
- Storage:
- Store at +4°C
- Molecular Formula:
- C35H42N4O6
- Molecular Weight (kDa):
- 614.73
- Soluble:
- DMSO
Description
- Description:
- Potent and selective CCK2 receptor antagonist
Biological Activity
- Biological Activity:
- CI 988 is a potent and selective CCK2 receptor antagonist. After oral administration, it exhibits anxiolytic activity.