Antalarmin hydrochloride

Antalarmin hydrochloride

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0155

CAS Number: 220953-69-5

Purity: ≥99% (HPLC)

Product Size Price
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Properties

  • Target:
  • CRF1 Receptor
  • CAS Number:
  • 220953-69-5
  • Chemical Name:
  • N-Butyl-N-ethyl-2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine hydrochloride
  • Storage:
  • Desiccate at +4°C
  • Molecular Formula:
  • C24H34N4.HCl
  • Molecular Weight (kDa):
  • 415.01
  • Soluble:
  • DMSO and Ethanol

Description

  • Description:
  • CRF1 receptor antagonist

Biological Activity

  • Biological Activity:
  • Antalarmin hydrochloride is a Corticotropin-Releasing hormone receptor 1 (CRF1) antagonist. It is a non-peptide antagonist and can suppress the secretion of ACTH induced by CRF.