Properties

• Target:
• CRF1 Receptor

• CAS Number:
• 257639-98-8

• Chemical Name:
• N-Butyl-N-ethyl-2,5-dimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine hydrochloride

• Storage:
• Desiccate at +4°C

• Molecular Formula:
• C23H32N4.HCl

• Molecular Weight (kDa):
• 400.99

• Soluble:
• DMSO and Ethanol

Description

• Description:
• Selective CRF1 receptor antagonist

Biological Activity

• Biological Activity:
• CP 154526 is a non-peptide selective Corticotropin-Releasing hormone receptor 1 (CRF1) antagonist. It is brain penetrant and displays anxiolytic-like activity.