BQ-123

BQ-123

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0185

CAS Number: 136553-81-6

Purity: ≥95% (HPLC)

Product Size Price
500 µg Online Inquiry

Properties

  • Target:
  • Endothelin ETA Receptor
  • CAS Number:
  • 136553-81-6
  • Storage:
  • Desiccate at -20°C
  • Molecular Formula:
  • C31H42N6O7
  • Molecular Weight (kDa):
  • 611
  • Soluble:
  • Water

Description

  • Description:
  • Selective ETA receptor antagonist

Biological Activity

  • Biological Activity:
  • BQ-123 is a endothelin-A (ETA) receptor antagonist. In rat model, it can reduce ventricular arrhythmias induced by ischemia.