G-15
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0206
CAS Number: 1161002-05-6
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- GPER
- CAS Number:
- 1161002-05-6
- Chemical Name:
- (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline
- Storage:
- Store at -20°C
- Molecular Formula:
- C19H16BrNO2
- Molecular Weight (kDa):
- 370.24
- Soluble:
- DMSO
Description
- Description:
- High affinity and selective GPER antagonist
Biological Activity
- Biological Activity:
- G-15 is a high affinity and selective GPER antagonist. It can inhibit calcium mobilization induced by agonist in vitro.