G-15

G-15

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0206

CAS Number: 1161002-05-6

Purity: ≥99% (HPLC)

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • GPER
  • CAS Number:
  • 1161002-05-6
  • Chemical Name:
  • (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline
  • Storage:
  • Store at -20°C
  • Molecular Formula:
  • C19H16BrNO2
  • Molecular Weight (kDa):
  • 370.24
  • Soluble:
  • DMSO

Description

  • Description:
  • High affinity and selective GPER antagonist

Biological Activity

  • Biological Activity:
  • G-15 is a high affinity and selective GPER antagonist. It can inhibit calcium mobilization induced by agonist in vitro.