GW 803430
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0228
CAS Number: 515141-51-2
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- MCH1 Receptor
- CAS Number:
- 515141-51-2
- Chemical Name:
- 6-(4-Chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3H)-one
- Storage:
- Store at +4°C
- Molecular Formula:
- C25H24ClN3O3S
- Molecular Weight (kDa):
- 481.99
- Soluble:
- HCl
Description
- Description:
- Selective MCH1 receptor antagonist
Biological Activity
- Biological Activity:
- GW 803430 is a selective melanin-concentrating hormone receptor 1 (MCH1 receptor) antagonist. It is orally active and displays antiobesity effects.