Properties

• Target:
• mGlu1 Receptor

• CAS Number:
• 869802-58-4

• Chemical Name:
• 9-(Dimethylamino)-3-(hexahydro-1H-azepin-1-yl)-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one

• Storage:
• Store at +4°C

• Molecular Formula:
• C17H21N5OS

• Molecular Weight (kDa):
• 343.45

• Soluble:
• DMSO

Description

• Description:
• Potent and selective mGluR1 receptor antagonist

Biological Activity

• Biological Activity:
• A 841720 is a potent and selective metabotropic glutamate receptor 1 (mGluR1) antagonist. It is non-conpetitive and demonstrats full efficacy in various animal pain models.