VU 0255035
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0257
CAS Number: 1135243-19-4
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- M1 Muscarinic Receptor
- CAS Number:
- 1135243-19-4
- Chemical Name:
- N-[3-Oxo-3-[4-(4-pyridinyl)-1-piperazinyl]propyl]-2,1,3-benzothiadiazole-4-sulfonamide
- Storage:
- Store at -20°C
- Molecular Formula:
- C18H20N6O3S2
- Molecular Weight (kDa):
- 432.52
- Soluble:
- DMSO
Description
- Description:
- Highly selective M1 muscarinic receptor antagonist
Biological Activity
- Biological Activity:
- VU 0255035 is a highly selective M1 muscarinic receptor antagonist. It is brain penetrant and can reduce pilocarpine-induced seizures in mice.