VU 0255035

VU 0255035

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0257

CAS Number: 1135243-19-4

Purity: ≥99% (HPLC)

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • M1 Muscarinic Receptor
  • CAS Number:
  • 1135243-19-4
  • Chemical Name:
  • N-[3-Oxo-3-[4-(4-pyridinyl)-1-piperazinyl]propyl]-2,1,3-benzothiadiazole-4-sulfonamide
  • Storage:
  • Store at -20°C
  • Molecular Formula:
  • C18H20N6O3S2
  • Molecular Weight (kDa):
  • 432.52
  • Soluble:
  • DMSO

Description

  • Description:
  • Highly selective M1 muscarinic receptor antagonist

Biological Activity

  • Biological Activity:
  • VU 0255035 is a highly selective M1 muscarinic receptor antagonist. It is brain penetrant and can reduce pilocarpine-induced seizures in mice.