J 104129 fumarate
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0260
CAS Number: 257603-40-0
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
Properties
- Target:
- M3 Muscarinic Receptor
- CAS Number:
- 257603-40-0
- Chemical Name:
- (αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-pentenyl)-4-piperidinyl]benzeneacetamide fumarate
- Storage:
- Store at +4°C
- Molecular Formula:
- C24H36N2O2.C4H4O4
- Molecular Weight (kDa):
- 500.63
- Soluble:
- DMSO and Ethanol
Description
- Description:
- Potent and selective M3 muscarinic receptor antagonist
Biological Activity
- Biological Activity:
- J 104129 fumarate is a potent and selective M3 muscarinic receptor antagonist. It can inhibit ACh-induced bronchoconstriction.