ML 154

ML 154

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0267

CAS Number: 1345964-89-7

Purity: 99%

Product Size Price
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Properties

  • Target:
  • NPS Receptor
  • CAS Number:
  • 1345964-89-7
  • Chemical Name:
  • 1-cinnamyl-3-(diphenylphosphorothioyl)-2-methyl-1H-imidazo[1,2-a]pyridin-4-ium bromide
  • Storage:
  • Store at -20°C
  • Molecular Formula:
  • C29H26N2PS.Br
  • Molecular Weight (kDa):
  • 545.47
  • Soluble:
  • DMSO

Description

  • Description:
  • Selective NPS receptor antagonist

Biological Activity

  • Biological Activity:
  • ML 154 is a selective neuropeptide S (NPS) receptor antagonist. It is competitive and brain penetrant. ML 154 can block NPS-induced ERK phosphorylation.