ML 154
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0267
CAS Number: 1345964-89-7
Purity: 99%
Product Size | Price |
---|---|
5 mg | Online Inquiry |
25 mg | Online Inquiry |
Properties
- Target:
- NPS Receptor
- CAS Number:
- 1345964-89-7
- Chemical Name:
- 1-cinnamyl-3-(diphenylphosphorothioyl)-2-methyl-1H-imidazo[1,2-a]pyridin-4-ium bromide
- Storage:
- Store at -20°C
- Molecular Formula:
- C29H26N2PS.Br
- Molecular Weight (kDa):
- 545.47
- Soluble:
- DMSO
Description
- Description:
- Selective NPS receptor antagonist
Biological Activity
- Biological Activity:
- ML 154 is a selective neuropeptide S (NPS) receptor antagonist. It is competitive and brain penetrant. ML 154 can block NPS-induced ERK phosphorylation.