BIIE 0246

BIIE 0246

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0270

CAS Number: 246146-55-4

Purity: ≥98% (HPLC)

Product Size Price
1 mg Online Inquiry
10 mg Online Inquiry

Properties

  • Target:
  • NPY Y2 Receptor
  • CAS Number:
  • 246146-55-4
  • Chemical Name:
  • N-[(1S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide
  • Storage:
  • Store at +4°C
  • Molecular Formula:
  • C49H57N11O6
  • Molecular Weight (kDa):
  • 896.06
  • Soluble:
  • DMSO and Ethanol

Description

  • Description:
  • Potent and selective NPY Y2 receptor antagonist

Biological Activity

  • Biological Activity:
  • BIIE 0246 is a potent and selective neurpeptide Y (NPY) Y2 receptor antagonist. It is a competitive antagonist and active in vivo.