BIIE 0246
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0270
CAS Number: 246146-55-4
Purity: ≥98% (HPLC)
Product Size | Price |
---|---|
1 mg | Online Inquiry |
10 mg | Online Inquiry |
Properties
- Target:
- NPY Y2 Receptor
- CAS Number:
- 246146-55-4
- Chemical Name:
- N-[(1S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide
- Storage:
- Store at +4°C
- Molecular Formula:
- C49H57N11O6
- Molecular Weight (kDa):
- 896.06
- Soluble:
- DMSO and Ethanol
Description
- Description:
- Potent and selective NPY Y2 receptor antagonist
Biological Activity
- Biological Activity:
- BIIE 0246 is a potent and selective neurpeptide Y (NPY) Y2 receptor antagonist. It is a competitive antagonist and active in vivo.