SR 142948
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0273
CAS Number: 184162-64-9
Purity: ≥97% (HPLC)
Product Size | Price |
---|---|
1 mg | Online Inquiry |
10 mg | Online Inquiry |
Properties
- Target:
- NTS Receptor
- CAS Number:
- 184162-64-9
- Chemical Name:
- 2-[[[5-(2,6-Dimethoxyphenyl)-1-[4-[[[3-(dimethylamino)propyl]methylamino]carbonyl]-2-(1-methylethyl)phenyl]-1H-pyrazol-3-yl]carbonyl]amino]-tricyclo[3.3.1.13,7]decane-2-carboxylic acid
- Storage:
- Store at +4°C
- Molecular Formula:
- C39H51N5O6
- Molecular Weight (kDa):
- 656.86
- Soluble:
- Water and DMSO
Description
- Description:
- Potent NTS receptor antagonist
Biological Activity
- Biological Activity:
- SR 142948 is a potent non-peptide neurotensin (NTS) receptor antagonist. It is orally active in vivo.