TCS1102
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0291
CAS Number: 916141-36-1
Purity: 98%
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- Orexin Receptor
- CAS Number:
- 916141-36-1
- Chemical Name:
- (S)-N-(Biphenyl-2-yl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide
- Storage:
- Store at RT
- Molecular Formula:
- C27H26N4O2S
- Molecular Weight (kDa):
- 470.59
- Soluble:
- DMSO
Description
- Description:
- Potent and selective dual orexin receptor antagonist
Biological Activity
- Biological Activity:
- TCS1102 is a potent and selective dual orexin receptor antagonist. It exihibits central activity in vivo.