Properties

• Target:
• OX₁ Receptor

• CAS Number:
• 1354039-86-3

• Chemical Name:
•  (aR,1S)-1-[(3,4-Dimethoxyphenyl)methyl]-3,4-dihydro-6,7-dimethoxy-N-(1-methylethyl)-a-phenyl-2(1H)-isoquinolineacetamide

• Storage:
• Store at +4°C

• Molecular Formula:
• C31H38N2O5

• Molecular Weight (kDa):
• 518.64

• Soluble:
• DMSO and Ethanol

Description

• Description:
• Potent and selective OX₁ receptor antagonist

Biological Activity

• Biological Activity:
• ACT 335827 is a potent and selective orexin OX₁ receptor antagonist. It is orally active and brain penetrant.