SB 674042
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0294
CAS Number: 483313-22-0
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- OX1 Receptor
- CAS Number:
- 483313-22-0
- Chemical Name:
- [5-(2-Fluorophenyl)-2-methyl-4-thiazolyl][2(S)-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl-1-pyrrolidinyl]methanone
- Storage:
- Store at +4°C
- Molecular Formula:
- C24H21FN4O2S
- Molecular Weight (kDa):
- 448.51
- Soluble:
- DMSO and Ethanol
Description
- Description:
- Potent and selective non-peptide OX1 receptor antagonist
Biological Activity
- Biological Activity:
- SB 674042 is a potent and selective non-peptide orexin OX1 receptor antagonist. It has no effect at dopaminergic, adrenergic, serotonergic, or purinergic receptors.