Properties

• Target:
• Prostaglandin E₄ Receptor

• CAS Number:
• 1155773-15-1

• Chemical Name:
• (S,Z)-1'-(3,5-Dimethylbenzyl)-2-ethyl-7,9-dimethoxy-10-methyl-5,10-dihydrospiro[benzo[e]imidazo[1,5-a]azepine-1,4'-piperidin]-3(2H)-one

• Storage:
• Store at +4°C

• Molecular Formula:
• C30H39N3O3

• Molecular Weight (kDa):
• 489.65

• Soluble:
• DMSO

Description

• Description:
• Highly selective PGE2 receptor EP4 antagonist

Biological Activity

• Biological Activity:
• ER-819762 is a highly selective prostanoid EP4 receptor antagonist. It has the potential for the treatment of chronic inflammatory pain.