L-161,982
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0314
CAS Number: 147776-06-5
Purity: ≥99% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
Properties
- Target:
- Prostaglandin E4 Receptor
- CAS Number:
- 147776-06-5
- Chemical Name:
- N-[[4'-[[3-Butyl-1,5-dihydro-5-oxo-1-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-4-yl]methyl][1,1'-biphenyl]-2-yl]sulfonyl]-3-methyl-2-thiophenecarboxamide
- Storage:
- Desiccate at +4°C
- Molecular Formula:
- C32H29F3N4O4S2
- Molecular Weight (kDa):
- 654.72
- Soluble:
- DMSO
Description
- Description:
- Selective EP4 receptor antagonist
Biological Activity
- Biological Activity:
- L-161,982 is a selective prostanoid EP4 receptor antagonist. It can suppresse bone formation induced by PGE2 in rats.