Properties

• Target:
• PAR1

• CAS Number:
• 474550-69-1

• Chemical Name:
• 1-(3-tert-butyl-4-methoxy-5-morpholinophenyl)-2-(5,6-diethoxy-7-fluoro-1-iminoisoindolin-2-yl)ethanone hydrobromide

• Storage:
• Store at +4°C

• Molecular Formula:
• C29H38FN3O5.HBr

• Molecular Weight (kDa):
• 608.54

• Soluble:
• DMSO

Description

• Description:
• Potent PAR1 antagonist

Biological Activity

• Biological Activity:
• E 5555 hydrobromide is a potent protease-activated receptor-1 (PAR1) antagonist. It is orally active and can inhibit thrombin-induced human platelet aggragation.