Properties

• Target:
• P2Y₂ Receptor

• CAS Number:
• 216657-60-2

• Chemical Name:
• 5-[[5-(2,8-Dimethyl-5H-dibenzo[a,d]cyclohepten-5-yl)-3,4-dihydro-2-oxo-4-thioxo-1(2H)-pyrimidinyl]methyl]-N-2H-tetrazol-5-yl-2-furancarboxamide

• Storage:
• Store at -20°C

• Molecular Formula:
• C28H23N7O3S

• Molecular Weight (kDa):
• 537.59

• Soluble:
• DMSO

Description

• Description:
• Selective, competitive P2Y₂ receptor antagonist

Biological Activity

• Biological Activity:
• AR-C 118925XX is a selectiv P2Y₂ antagonist. It is a competitive antagonist and can inhibit the translocation of β-arrestin induced by P2Y₂ receptor in vitro.