Properties

• Target:
• NK1 Receptor

• CAS Number:
• 414910-30-8

• Chemical Name:
• (2R,4S)-4-(4-acetylpiperazin-1-yl)-N-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethyl)-2-(4-fluoro-2-methylphenyl)-N-methylpiperidine-1-carboxamide methanesulfonate

• Storage:
• Store at -20°C

• Molecular Formula:
• C30H35F7N4O2.CH4O3S

• Molecular Weight (kDa):
• 712.72

• Soluble:
• Water and DMSO

Description

• Description:
• Potent and selective NK1 receptor antagonist

Biological Activity

• Biological Activity:
• Casopitant mesylate is a potent and selective neurokinin 1 (NK1) receptor antagonist. It is orally active.