Properties

• Target:
• NK2 Receptor

• CAS Number:
• 158848-32-9

• Chemical Name:
• 5-Fluoro-3-[2-[4-methoxy-4-[[(R)-phenylsulphinyl]methyl]-1-piperidinyl]ethyl]-1H-indole

• Storage:
• Desiccate at -20°C

• Molecular Formula:
• C23H27FN2O2S

• Molecular Weight (kDa):
• 414.54

• Soluble:
• DMSO and Ethanol

Description

• Description:
• Potent and selective NK2 receptor antagonist

Biological Activity

• Biological Activity:
• GR 159897 is a potent and selective neurokinin 2 (NK2) receptor antagonist. It is a non-peptide and orally active antagonist.GR 159897 exerts anxiolytic activity in vivo.