SB 657510
For Research Use Only. Not For Clinical Use.
Catalog Number: ANG0367
CAS Number: 474960-44-6
Purity: ≥98% (HPLC)
Product Size | Price |
---|---|
10 mg | Online Inquiry |
50 mg | Online Inquiry |
Properties
- Target:
- Urotensin-ⅡReceptor
- CAS Number:
- 474960-44-6
- Chemical Name:
- 2-Bromo-N-[4-chloro-3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]phenyl]-4,5-dimethoxybenzenesulfonamide
- Storage:
- Store at RT
- Molecular Formula:
- C19H22BrClN2O5S
- Molecular Weight (kDa):
- 505.81
- Soluble:
- DMSO
Description
- Description:
- Selective urotensin-Ⅱ receptor antagonist
Biological Activity
- Biological Activity:
- SB 657510 is a selective urotensin-Ⅱ receptor antagonist. It can Inhibit the intracellular Ca2+ mobilization induced by urotensin-Ⅱ.