SB 657510

SB 657510

For Research Use Only. Not For Clinical Use.

Catalog Number: ANG0367

CAS Number: 474960-44-6

Purity: ≥98% (HPLC)

Product Size Price
10 mg Online Inquiry
50 mg Online Inquiry

Properties

  • Target:
  • Urotensin-ⅡReceptor
  • CAS Number:
  • 474960-44-6
  • Chemical Name:
  • 2-Bromo-N-[4-chloro-3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]phenyl]-4,5-dimethoxybenzenesulfonamide
  • Storage:
  • Store at RT
  • Molecular Formula:
  • C19H22BrClN2O5S
  • Molecular Weight (kDa):
  • 505.81
  • Soluble:
  • DMSO

Description

  • Description:
  • Selective urotensin-Ⅱ receptor antagonist

Biological Activity

  • Biological Activity:
  • SB 657510 is a selective urotensin-Ⅱ receptor antagonist. It can Inhibit the intracellular Ca2+ mobilization induced by urotensin-Ⅱ.