Properties

• Target:
• Vasopressin V1a Receptor

• CAS Number:
• 150375-75-0

• Chemical Name:
• (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide

• Storage:
• Store at +4°C

• Molecular Formula:
• C28H27Cl2N3O7S

• Molecular Weight (kDa):
• 620.5

• Soluble:
• DMSO

Description

• Description:
• Potent and selective vasopressin V1a receptor antagonist

Biological Activity

• Biological Activity:
• SR 49059 is a potent and selective vasopressin V1a receptor antagonist. It is orally active and can antagonize arginine vasopressin-induced effects in vitro.